Archived: 6th Winter Conference
on Medicinal & Bioorganic Chemistry

The Viagra Story

The Kaletra-Ritonavir Story

The Neurontin Story

Reagents in Organic Synthesis: The Discovery and the Early Years

Transition Metal Catalyzed Sequential Coupling via C-H Bond Cleavage

Concepts of Nature in Organic Synthesis: Cascade Catalysis and Multistep Conversions in Concert

Tandem and Cascade Carbon-Carbon Bond-Forming Processes Catalyzed by Pd and Zr Complexes

Soluble Polymers as Easily Separable Supports in Synthesis and Catalysis

ROM-Polymerization Strategies for Facilitated Synthesis

Development of New Methods for Organic Synthesis

Polymer-Assisted Solution-Phase (PASP) Chemical Library Synthesis and its Application on the Tissue Factor VIIa Projects

Benzopyrans are selective ERbagonists for use in the treatment of prostatic diseases

Design and Development of Low Toxicity UAB-rexinoids for Breast Cancer Chemoprevention

In vitro and In vivo of a ketone-containing a_vb₃ integrin antagonist for the treatment for osteoporosis

Computational and Pharmacokinetic Studies Directed at Understanding the Differences in Oral Bioavailability Seen between Closely Related a_Vb₃integrin Antagonists

Synthesis of Immunomodulatory Macrolides for Cystic Fibrosis

Progression of a Novel Class of Orally Active p38 Map Kinase Inhibitors

Synthesis and Modelling Studies of Peptidomimetic Aldehydes Related to a Cataract Preventing Calpain Inhibitor

Structure-based design of a series of potent and selective cell permeable inhibitors of humanb–secretase

Drug Discovery at Adaptive Signaling Interfaces

Dallas Binding Sites and Conformational Changes in Protein Kinases

Exploiting Plasticity in Nuclear Receptor Drug Discovery

Targeting Protein-Protein and Protein-DNA Interaction using Solution Phase Combinatorial Chemistry

The Poisoning of Human Topoisomerase I by Structurally Diverse Anticancer Compounds and Various Insults to DNA

Challenges for Drug Discovery at Protein/Protein Interfaces

Starting Small and Strong: Fragment Based Drug Discovery

Development of a Potent HIV-1 Integrase Inhibitor with a Unique Resistance Profile

Double Oxidation of Tryptophanes: Synthesis of the Potent Anthelmintic Pyrrolobenzoxazine CJ-12662¹

Calcitonin gene-related peptide antagonists

APD 356, A Potent and Selective 5HT_2C Agonist is a Potential New Treatment for Obesity

Diagnostics Structure-based Optimization of Novel Azepane Derivatives as PKB Selective Inhibitors

Identification and Development of Potent and Selective P13Kỷ Inhibitors

Unusual Heterocycle Synthesis: Routes to Pyrazolo[1,5-a]Pyridine Compounds as P38 Kinase Inhibitors